CB1-IN-1 Catalog No.:M21313-C but has minimal effect on

but has minimal effect on viability of nontransformed human cells

and 50 mg/ kg)

CAS Number: 38927-54-7

Potassium canrenoate

Smiles: NCCOCCOC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O

CB1-IN-1 Catalog No.:M21313-C but has minimal effect onCB1 IN 1 (BPRCB1184) is a peripherally restricted CB1R antagonist, with Ki of 0. 3 nM and 21 nM for CB1R (EC50 = 3 nM) and CB2R, respectively. IC50 value: 0. 3 nM (Ki, CB1R) 21 nM (Ki, CB2R)Target: CB1Rin vivo: CB1 IN 1 is a novel peripherally restricted cannabinoid 1 receptor antagonist with significant weight loss efficacy in diet induced obese mice. CB1 IN 1 has great potential to ameliorate this related metabolic syndrome. Product information CAS